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Search Results for " σ1 receptor antagonist-1 "

9

Compounds

Cat No. Product Name Synonyms Targets
T9244 σ1 Receptor antagonist-1 Sigma receptor
σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.
T12911 Sigma-1 receptor antagonist 2 Sigma receptor
Sigma-1 receptor antagonist 2 is a potent and selective antagonist of sigma 1 receptor (σ1 R) (σ1 and σ2 receptor with Kis of 3.88 and 1288 nM , respectively).
T12912 Sigma-1 receptor antagonist 3 Sigma receptor , HER
Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain.
T7488 BD1063 dhydrochloride BD1063 Sigma receptor
BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).
T8834 EST64454 hydrochloride EST64454 Sigma receptor
EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.
T21788 BD 1008 dihydrobromide Sigma receptor
BD 1008 dihydrobromide is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM). BD 1008 dihydrobromide have high affinity for sigma1 receptors, moderate affinity for sigma2 receptors.
T61901 σ1 Receptor/μ Opioid receptor modulator 1
σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM). Opioid receptor modulator 1 shows potent analgesic activity, and ...
T9669 EST73502 hydrochloride
EST73502 hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with K i s of 64 nM and 118 nM for MOR and σ1R, respecti...
T39176 PB28
PB28 is a cyclohexylpiperazine derivative that functions as a potent and highly selective agonist of the sigma 2 (σ2) receptor, exhibiting a Ki (binding affinity) of 0.68 nM. At the same time, PB28 acts as an antagonist ...
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